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SotA/Medical/Single-step retrosynthesis/USPTO-50k

Single-step retrosynthesis on USPTO-50k

Metric: Top-5 accuracy (higher is better)

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Results

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#Model↕Top-5 accuracy▼Extra DataPaperDate↕Code
1O-GNN (reaction class as prior)93.4No--Code
2LocalRetro (reaction class as prior)92.4No--Code
3UAlign (reaction class as prior)91.5NoUAlign: Pushing the Limit of Template-free Retro...2024-03-25Code
4NAG2G (reaction class as prior)90.5NoNode-Aligned Graph-to-Graph (NAG2G): Elevating T...2023-09-27Code
5MARS (reaction class as prior)90.2NoMARS: A Motif-based Autoregressive Model for Ret...2022-09-27-
6SemiRetro (reaction class as prior)89.8NoSemiRetro: Semi-template framework boosts deep r...2022-02-12-
7RetroComposer (reaction class as prior)89.5NoRetroComposer: Composing Templates for Template-...2021-12-20Code
8MEGAN (reaction class as prior)87.5NoMolecule Edit Graph Attention Network: Modeling ...2020-06-27Code
9O-GNN (reaction class unknown)86No--Code
10LocalRetro (reaction class unknown)85.9No--Code
11GraphRetro (reaction class as prior)85.2NoLearning Graph Models for Retrosynthesis Predict...2020-06-12-
12Dual-TF (reaction class as prior)84.7NoEnergy-based View of Retrosynthesis2020-07-14-
13UAlign (reaction class unknown)84.6NoUAlign: Pushing the Limit of Template-free Retro...2024-03-25Code
14NAG2G (reaction class unknown)83.4NoNode-Aligned Graph-to-Graph (NAG2G): Elevating T...2023-09-27Code
15MARS (reaction class unknown)83.3NoMARS: A Motif-based Autoregressive Model for Ret...2022-09-27-
16RetroComposer (reaction class unknown)83.2NoRetroComposer: Composing Templates for Template-...2021-12-20Code
17RetroSim (reaction class as prior)81.2No--Code
18MHNreact (reaction class unknown)81.2No--Code
19Augmented Transformer (reaction class unknown)81NoState-of-the-Art Augmented NLP Transformer model...2020-03-05Code
20SemiRetro (reaction class unknown)80.4NoSemiRetro: Semi-template framework boosts deep r...2022-02-12-
21MEGAN (reaction class unknown)78.4NoMolecule Edit Graph Attention Network: Modeling ...2020-06-27Code
22GLN75.6NoRetrosynthesis Prediction with Conditional Graph...2020-01-06Code
23GET-LT1 (reaction class as prior)74.8No---
24Dual-TF (reaction class unknown)74.6NoEnergy-based View of Retrosynthesis2020-07-14-
25G2GT (reaction class unknown)74.5NoG2GT: Retrosynthesis Prediction with Graph to Gr...2022-04-19Code
26RetroPrime (reaction class unknown)74No--Code
27GET-LT2 (reaction class as prior)72.5No---
28G2Gs72.5NoA Graph to Graphs Framework for Retrosynthesis P...2020-03-28-
29GraphRetro (reaction class unknown)72.2NoLearning Graph Models for Retrosynthesis Predict...2020-06-12-
30Graph2SMILES-D-GAT (reaction class unknown)70.4NoPermutation invariant graph-to-sequence model fo...2021-10-19Code
31Graph2SMILES-D-GCN (reaction class unknown)70NoPermutation invariant graph-to-sequence model fo...2021-10-19Code
32RetroSim (reaction class unknown)63.3No--Code
33GET-LT1 (reaction class unknown)62.4No---
34Chemformer-Large (reaction class unknown)62.3No--Code
35Expert System (reaction class as prior)59.1NoRetrosynthetic reaction prediction using neural ...2017-06-06Code