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SotA/Medical/Single-step retrosynthesis/USPTO-50k

Single-step retrosynthesis on USPTO-50k

Metric: Top-3 accuracy (higher is better)

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Results

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#Model↕Top-3 accuracy▼Extra DataPaperDate↕Code
1O-GNN (reaction class as prior)87.7No--Code
2UAlign (reaction class as prior)86.7NoUAlign: Pushing the Limit of Template-free Retro...2024-03-25Code
3NAG2G (reaction class as prior)86.4NoNode-Aligned Graph-to-Graph (NAG2G): Elevating T...2023-09-27Code
4LocalRetro (reaction class as prior)86.1No--Code
5MARS (reaction class as prior)85.8NoMARS: A Motif-based Autoregressive Model for Ret...2022-09-27-
6RetroComposer (reaction class as prior)85.8NoRetroComposer: Composing Templates for Template-...2021-12-20Code
7SemiRetro (reaction class as prior)85.7NoSemiRetro: Semi-template framework boosts deep r...2022-02-12-
8MEGAN (reaction class as prior)82NoMolecule Edit Graph Attention Network: Modeling ...2020-06-27Code
9Dual-TF (reaction class as prior)81.9NoEnergy-based View of Retrosynthesis2020-07-14-
10GraphRetro (reaction class as prior)81.5NoLearning Graph Models for Retrosynthesis Predict...2020-06-12-
11O-GNN (reaction class unknown)77.7No--Code
12LocalRetro (reaction class unknown)77.5No--Code
13UAlign (reaction class unknown)77.3NoUAlign: Pushing the Limit of Template-free Retro...2024-03-25Code
14RetroComposer (reaction class unknown)77.2NoRetroComposer: Composing Templates for Template-...2021-12-20Code
15NAG2G (reaction class unknown)76.9NoNode-Aligned Graph-to-Graph (NAG2G): Elevating T...2023-09-27Code
16MARS (reaction class unknown)76.4NoMARS: A Motif-based Autoregressive Model for Ret...2022-09-27-
17SemiRetro (reaction class unknown)75.3NoSemiRetro: Semi-template framework boosts deep r...2022-02-12-
18MHNreact (reaction class unknown)74.6No--Code
19RetroSim (reaction class as prior)73.8No--Code
20GET-LT1 (reaction class as prior)71.3No---
21RetroPrime (reaction class unknown)70.8No--Code
22Dual-TF (reaction class unknown)70.7NoEnergy-based View of Retrosynthesis2020-07-14-
23MEGAN (reaction class unknown)70.7NoMolecule Edit Graph Attention Network: Modeling ...2020-06-27Code
24G2GT (reaction class unknown)69.9NoG2GT: Retrosynthesis Prediction with Graph to Gr...2022-04-19Code
25GET-LT2 (reaction class as prior)69.4No---
26GLN69NoRetrosynthesis Prediction with Conditional Graph...2020-01-06Code
27GraphRetro (reaction class unknown)68.3NoLearning Graph Models for Retrosynthesis Predict...2020-06-12-
28G2Gs67.6NoA Graph to Graphs Framework for Retrosynthesis P...2020-03-28-
29Graph2SMILES-D-GCN (reaction class unknown)66.5NoPermutation invariant graph-to-sequence model fo...2021-10-19Code
30Graph2SMILES-D-GAT (reaction class unknown)66.3NoPermutation invariant graph-to-sequence model fo...2021-10-19Code
31GET-LT1 (reaction class unknown)58.8No---
32RetroSim (reaction class unknown)54.7No--Code
33Expert System (reaction class as prior)52.3NoRetrosynthetic reaction prediction using neural ...2017-06-06Code